EMD-44635
Inactive mu opioid receptor bound to Nb6, naloxone and NAM
EMD-44635
Single-particle3.26 Å
![EMD-44635](https://cdn.statically.io/img/www.ebi.ac.uk/emdb/images/entry/EMD-44635/400_44635.gif)
Map released: 17/07/2024
Last modified: 24/07/2024
Sample Organism:
Mus musculus,
Lama glama
Sample: mu-type opioid receptor with kappa-type opioid receptor ICL3 in complex with Nb6, naloxone and a negative allosteric modulator
Fitted models: 9bjk
Deposition Authors: O'Brien ES
,
Wang H,
Kaavya Krishna K,
Zhang C,
Kobilka BK
Sample: mu-type opioid receptor with kappa-type opioid receptor ICL3 in complex with Nb6, naloxone and a negative allosteric modulator
Fitted models: 9bjk
Deposition Authors: O'Brien ES
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A mu-opioid receptor modulator that works cooperatively with naloxone.
O'Brien ES
,
Rangari VA
,
El Daibani A,
Eans SO,
Hammond HR,
White E,
Wang H,
Shiimura Y,
Krishna Kumar K
,
Jiang Q,
Appourchaux K
,
Huang W,
Zhang C,
Kennedy BJ
,
Mathiesen JM,
Che T
,
McLaughlin JP
,
Majumdar S
,
Kobilka BK
(2024) Nature , 631 , 686 - 693
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(2024) Nature , 631 , 686 - 693